Dr Sandeep Chandrashekharappa
Assistant Professor
| Department of Medicinal Chemistry
National Institute of Pharmaceutical Education and Research, Raebareli
Uttar Pradesh
Expertise:
Organic Chemistry
167
Publications
8
Projects
2547
Scopus Citations
2261
CrossRef
19 Years 5 Months Total Experience
Scopus
2,547
Citations
30
h-index
CrossRef
2,261
Citations
28
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Professional Recognition
Gandian Young Technological innovation award
2019
Govt of India
Star Award
2011
BBRC Bangalore
Star Award
2012
BBRC Bangalore
Bridging Postdoctoral Fellowship
2015
Instem Bangalore
Gnanoday Puraskar
2025
NIPER raebareli
Community & Membership
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Personal Details
Doctor of Philosophy
2014
Phytosynthese
Master of Science
2005
Phytosynthese
Assistant Professor
Mar 2021 – Present
National Institute of Pharmaceutical Education and Research, Raebareli
| Department of Medicinal Chemistry
Post-Doctoral Fellow
Sep 2015 – Mar 2021
INSTITUTE OF
Associate Scientist
Aug 2005 – Dec 2013
Biocon BMS Research Centre
Chemical Sciences
Scholarly Work
Developing technologies to decontaminate pesticides/insecticides in spices
OtherLead optimization of sulfone, efloxate and adamantyl urea derivatives against drug-resistant M. tuberculosis
OtherAdamantyl Urea Derivatives as Mmpl3 Inhibitors: A New Avenue for the Treatment of Drug-Resistant Tuberculosis
OtherSynthesis and Evaluation of Nitrogen Tethered Derivatives in Cell-Based and Animal Models of Acute Lung Injury
OtherSynthesis, safety and efficacy of aminobutyric acid linked curcumin nanodiamond conjugate for the treatment of Alzheimer's disease
OtherDevelopment and Evaluation of Novel Multi-Target Urolithin Analogues as Potential Neuroprotective Therapeutics for Ischemic Stroke
CompletedDesign, synthesis, characterization of Dibromo Indolizine analogs and evaluation of their anti-inflammatory activity in lipopolysaccharide (LPS)-induced model in vitro
OtherProphylactic catalytic dermal cream to prevent pesticide exposure during farming practices
CompletedNo Data Found
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A One-pot Process For Preparation Of 2-substituted-1H-benzo[d]imidazole Derivatives
NIPER Raebareli
-
Patent No. :
557854
Filed :
28-06-2024
Published :
13-01-2025
Granted
(E)-1-(2-(4-substituedphenyl)-2-oxoethyl)-4-((hydroxyimino)methyl)pyridinium bromides as anti-tubercular agents
KFU
-
Patent No. :
US patent Pub No: US 12, 215, 082 B1
Filed :
26-06-2024
Published :
04-02-2025
Granted
A PROCESS FOR SYNTHESIS OF CHROMONE AND FLAVONE AND THEIR USE IN PHARMACEUTICAL APPLICATIONS
NIPER Raebareli
-
Patent No. :
557480
Filed :
30-03-2024
Published :
06-01-2025
Granted
Novel benzofuro[2,3-c]pyridinol compounds and process for preparation thereof
NIPER Raebareli
-
Patent No. :
569870
Filed :
19-03-2024
Published :
19-08-2025
Granted
A PROCESS FOR PREPARATION OF BENZOFURAN AND BENZOFURO[2,3-C]PYRIDINE COMPOUNDS
NIPER Raebareli
-
Patent No. :
552392
Filed :
11-03-2024
Published :
15-10-2024
Granted
Pyrrolo[1,2-a] imidazole, 1H-Pyrrole-3-carboxylate analogues and process for preparation thereof
NIPER Raebareli
-
Patent No. :
553787
Filed :
21-02-2024
Published :
01-11-2024
Granted
Development of (E)-3-(substitutedbenzoyl)-7-((hydroxyimino)methyl)-2-substitutedindolizine-1-carboxylate derivatives as anti-tubercular agents
Katharigatta N. Venugopala
Sandeep Chandrashekharappa
Melendran Pillay
Pran Kishore Deb
Rashmi Venugopala
Viresh Mohanlall
-
Application No. :
18/531,129
Filed :
06-12-2023
Published :
30-11--0001
Filed
(E)-1-(2-(4-substituedphenyl)-2-oxoethyl)-4-((hydroxyimino)methyl)pyridinium bromides as anti-tubercular agents.
Katharigatta N. Venugopala
Sandeep Chandrashekharappa
Melendran Pillay
Pran Kishore Deb
Rashmi Venugopala
-
Application No. :
18386017
Filed :
23-11-2023
Published :
30-11--0001
Filed
Adenosine receptor activity of substituted benzoyl-7-methoxyindolizine-1-carboxylate analogues
Katharigatta N. Venugopala
Rahul D. Nagdeve
Pran Kishore Deb
Buccioni Michela
Gabriella Marucci
Susanta K. Nayak
Sandeep Chandrashekharappa
Osama I. Alwassil
Rashmi Venugopala
-
Application No. :
18386397
Filed :
02-11-2023
Published :
30-11--0001
Filed
7-Isopropyl 1-ethyl/methyl 3-(substituted benzoyl)-2-substituted indolizine-1,7-dicarboxylates as larvicidal agents
Katharigatta N. Venugopala
Sandeep Chandrashekharappa
Pran Kishore Deb
Osama I. Alwassil
Rashmi Venugopala.
-
Application No. :
18/500,084,
Filed :
01-11-2023
Published :
30-11--0001
Filed
Substituted 7-amino-3-(substituted benzoyl)indolizine-1-carboxylates as anti-tubercular agents.
Katharigatta N. Venugopala
Melendran Pillay
Vijaykumar Uppar
Pran Kishore Deb
Rashmi Venugopala
Sandeep Chandrashekharappa
Basavaraj Padmashali
-
Application No. :
18382829
Filed :
23-10-2023
Published :
30-11--0001
Filed
Ethyl-1-(substitutedbenzoyl)-5-methylpyrrolo [1, 2-a] quinoline-3-carboxylates as anticancer agents
Katharigatta N. Venugopala
Vijaykumar Uppar
Rashmi Venugopala
Sandeep Chandrashekharappa
Basavaraj Padmashali
Viresh Mohanlall.
-
Patent No. :
US Patent 12,194,029,
Filed :
23-10-2023
Published :
14-01-2025
Granted
4-Cyano-1-(2-oxo-2-(substituted phenyl)ethyl)pyridin-1-ium bromides as anti-tubercular agents
Katharigatta N. Venugopala
Mohamed A. Morsy
Sandeep Chandrashekharappa
Melendran Pillay.
-
Patent No. :
US 12, 202, 801 B1
Filed :
23-10-2023
Published :
21-01-2025
Granted
(2-(SUBSTITUTED PHENYL)-2- OXOE- THYL)- 4-METHYLPYRIDIN-1-IUM BRO- MIDE AS ANTI-TUBERCULAR AGENTS
KFU
-
Patent No. :
US 12, 227, 480 B1
Filed :
23-10-2023
Published :
18-02-2025
Granted
Katharigatta N. Venugopala
Pran Kishore Deb
Mohamed A. Morsy
Bandar E. Aldhubiab
Sandeep Chandrashekharappa
Melendran Pillay.
-
Application No. :
Production of 1-(2-(substituted phenyl)-2-oxoethyl)-4-(isopropoxycarbonyl)pyridin-1-ium br
Filed :
10-10-2023
Published :
30-11--0001
Filed
(6-Methyl-4-substitutedphenyl-2-oxo/thioxo-1,2,3,4-tetrahydropyrimidin-5-yl)(piperidin-1-yl)methanones as anti-tubercular agents
Katharigatta N. Venugopala
Mohamed A. Morsy
Keshab M. Bairagi
Susanta K. Nayak
Melendran Pillay
Pran Kishore Deb
Sandeep Chandrashekharappa
Osama I. Alwassil
-
Application No. :
18367645
Filed :
13-09-2023
Published :
30-11--0001
Filed
(6-Methyl-4-substitutedphenyl-2-oxo/thioxo-1,2,3,4-tetrahydropyrimidin-5-yl)(piperidin-1-yl)methanones as anti-tubercular agents
Katharigatta N. Venugopala
Mohamed A. Morsy
Keshab M. Bairagi
Susanta K. Nayak
Melendran Pillay
Pran Kishore Deb
Sandeep Chandrashekharappa
Osama I. Alwassil
-
Application No. :
18367635
Filed :
13-09-2023
Published :
30-11--0001
Filed
Substituted 7-methyl quinoline derivatives as anti-tubercular agents.
Katharigatta N. Venugopala
Pran Kishore Deb
Melendran Pillay
Vijaykumar Uppar
Mohamed A. Morsy
Bandar E. Aldhubiab
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Sandeep Chandrashekharappa
Basavaraj Padmashali.
-
Application No. :
18240256
Filed :
30-08-2023
Published :
30-11--0001
Filed
Ethyl 2-substitued-1-(substitutedbenzoyl)-7-methylpyrrolo[1,2-a]quinoline-3-carboxylates as anti-tubercular agents.
Katharigatta N. Venugopala
Pran Kishore Deb
Melendran Pillay
Sandeep Chandrashekharappa
Mohamed A. Morsy
Bandar E. Aldhubiab
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Christophe Tratrat
Sheena Shashikanth
Vijaykumar Uppar
Basavaraj Padmashali.
-
Application No. :
18237273
Filed :
23-08-2023
Published :
30-11--0001
Filed
Ethyl 2-substitued-1-(substitutedbenzoyl)-7-methylpyrrolo[1,2-a]quinoline-3-carboxylates as anti-tubercular agents.
Katharigatta N. Venugopala
Pran Kishore Deb
Melendran Pillay
Sandeep Chandrashekharappa
Mohamed A. Morsy
Bandar E. Aldhubiab
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Christophe Tratrat
Sheena Shashikanth
Vijaykumar Uppar
Basavaraj Padmashali.
-
Patent No. :
US Patent 11,845,746, 2023
Filed :
23-08-2023
Published :
19-12-2023
Granted
1-Substitutedbenzoyl-4-bromopyrrolo[1,2-a]quinoline-3-carboxylate derivatives as anti-tubercular agents
Katharigatta N. Venugopala
Pran Kishore Deb
Melendran Pillay
Sandeep Chandrashekharappa
Mohamed A. Morsy
Bandar E. Aldhubiab
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Vijaykumar Uppar
Raghu Prasad Mailavaram
Basavaraj Padmashali.
-
Application No. :
18236237
Filed :
21-08-2023
Published :
30-11--0001
Filed
Adenosine receptor activity of methyl/ethyl 3-(substituted benzoyl)-6,8-dimethylindolizine-2-substituted-1-carboxylates
Katharigatta N. Venugopala
Buccioni Michela
Gabriella Marucci
Pran Kishore Deb
Mohamed A. Morsy
Bandar E. Aldhubiab
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Sandeep Chandrashekharappa
Sheena Shashikanth.
-
Application No. :
18230585
Filed :
08-08-2023
Published :
30-11--0001
Filed
Novel substituted phenyl quinolin-1-ium bromide derivative as antitubercular agents.
Katharigatta N. Venugopala
Pran Kishore Deb
Melendran Pillay
Sandeep Chandrashekharappa
Mohamed A. Morsy
Bandar E. Aldhubiab
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Christophe Tratrat
Sheena Shashikanth
-
Application No. :
18229825
Filed :
03-08-2023
Published :
30-11--0001
Filed
7-Isopropyl 1-ethyl/methyl 3-(substituted benzoyl)-2-substituted indolizine-1,7-dicarboxylates as anti-tubercular agents
Katharigatta N. Venugopala
Bandar E. Aldhubiab
Mohamed A. Morsy
Mahesh Attimarad
Anroop B. Nair
Nagaraja Sreeharsha
Christophe Tratrat
Sandeep Chandrashekharappa
Melendran Pillay
Pran Kishore Deb
Sheena Shashikanth
-
Application No. :
18191407
Filed :
30-03-2023
Published :
30-11--0001
Filed
ANTI-TB NAPHTHYRIDINE DERIVATIVES AND THEIR SYNTHESIS THEREOF
Ningegowda
Raghu; Savitha H S
Neethu Patil; Chandrashekharappa
Sandeep
-
Patent No. :
202341021764
Filed :
26-03-2023
Published :
31-03-2023
Filed
METHOD FOR SYNTHESIS OF CHRYSIN, TECTOCHRYSIN AND THEIR DERIVATIVES THEREOF FOR USE IN PHARMACEUTICAL APPLICATIONS
Niper Raebareli
-
Patent No. :
202211047585
Filed :
22-08-2022
Published :
30-11--0001
Filed
Antitubercular compounds
Katharigatta N Venugopala
Mahesh Attimarad
Anroop B Nair
Nagaraja Sreeharsha
Mohamed A Morsy
Sandeep Chandrashekharappa
Melendran Pillay
Pran Kishore Deb
-
Patent No. :
11530217
Filed :
29-06-2022
Published :
20-12-2022
Published
Compositions, materials, and methods for deactivating toxic agents;
InStem Bangalore
-
Patent No. :
IN 202142053063 A
Filed :
18-11-2021
Published :
10-12-2021
Published
N-(4-fluorophenyl)-5-phenyl-[1,2,4] triazolo [1,5-a] pyridine-2-carboxamide derivatives and their synthesis thereof
Ningegowda
Raghu; Banuprakash
Govindappa; Chandrashekharappa
Sandeep
-
Patent No. :
WO 2021161084 A1
Filed :
19-08-2021
Published :
30-11--0001
Published
Synthesis and characterization of (s)-3-(5-fluoropyridin-2-yl)-5-(piperidin-3-yl)-1,2,4-oxadiazole derivatives and their secretary phospholipase a2 (spla2) inhibitor activity
Ranjith Siddaraj
Raghu Ningegowda
Govindappa Banuprakash
Sandeep Chandrashekharappa
-
Patent No. :
WO 2022069953
Filed :
27-03-2021
Published :
07-04-2022
Published
Urolithin a and derivatives thereof for use in therapy
Jala
Venkatakrishna Rao; Bodduluri
Haribabu; Singh
Rajbir; Vemula
Praveen Kumar; Chandrashekharappa
Sandeep; Hiwale
Ankita Arun
-
Patent No. :
IN 202017054042 A
Filed :
26-02-2021
Published :
30-11--0001
Published
Synthesis and characterization of (s)-3-(5-fluoropyridin-2-yl)-5-(piperidin-3-yl)-1,2,4-oxadiazole derivatives and their secretary phospholipase a2 (spla2) inhibitor activity
Ranjith Siddaraj
Raghu Ningegowda
Govindappa Banuprakash
Sandeep Chandrashekharappa
-
Patent No. :
457614
Filed :
29-09-2020
Published :
23-04-2021
Published
Ethyl and dimethyl 1-benzoylpyrrolo [1,2-a] quinoline-3-carboxylate analog derivatives as antifungal and antibacterial agents
Basavaraj Padmashali
Vijayakumar Uppar
. Sandeep Chandrashekharappa
Kiran K. MudnakuduNagaraju
-
Patent No. :
394853
Filed :
12-08-2019
Published :
05-02-2021
Granted
Compounds, compositions, methods of using and methods for preparing comopunds
Jala VR
Bodduluri H
Singh R
Vemula PK
Chandrashekharappa S
Hiwale AA
-
Patent No. :
US 2021/0267932 A1
Filed :
14-05-2019
Published :
02-09-2021
Published
Compositions, materials, and methods for deactivating toxic agents
InStem Bangalore
-
Patent No. :
20419
Filed :
21-03-2019
Published :
30-11--0001
Filed
Treatment of Tuberculosis
Katharigatta N. Venugopala
Sandeep Chandrashekharappa
Pillay Melendhran
Bharti Odhav
Mohanlall Viresh
Kasumbwe kabange
-
Patent No. :
ZA 2020003088 A
Filed :
19-03-2019
Published :
30-06-2021
Published
Eco-friendly synthesis of pyrrolo [1,2-a] quinoline-3-carboxylate derivatives & their study of antibacterial and antioxidant properties
Vijayakumar Uppar
Basavaraj Padmashali
Govindappa Banuprakash
and Sandeep Chandrashekharappa
-
Patent No. :
418528
Filed :
12-02-2019
Published :
13-03-2020
Granted
N-(4-fluorophenyl)-5-phenyl-[1,2,4] triazolo [1,5-a] pyridine-2-carboxamide derivatives and their synthesis thereof
Raghu Ningegowda
Sandeep Chandrashekharappa
Govindappa Banuprakash
-
Patent No. :
399540
Filed :
21-01-2019
Published :
20-06-2022
Published
Novel Substituted Indolizine Scaffolds For MDR Strains OF Mycobacterium Tuberculosis, Synthetic Methodology And Chemical Structures Thereof
Sandeep Chandrashekharappa. Katharigatta N. Venugopala.
-
Patent No. :
IN 201941002546 A
Filed :
21-01-2019
Published :
03-04-2020
Published
Synthetic analogs of gut microbial metabolites for protection of endothelial and epithelial barriers and applications thereof
Jala VR
Bodduluri H
Singh R
Vemula PK
Chandrashekharappa S
Hiwale AA
-
Patent No. :
11202011261P
Filed :
15-05-2018
Published :
30-12-2020
Published
Urolithin a and derivatives thereof for use in therapy
InStem Bangalore
-
Patent No. :
WO 2019222146
Filed :
14-03-2018
Published :
21-11-2019
Published
Compositions, materials, and methods for deactivating toxic agents
InStem Bangalore
-
Patent No. :
WO 2019180653 A1
Filed :
13-02-2018
Published :
26-09-2019
Published
A conjugate, a composition, an article, processes of preparation and application thereof
InStem Bangalore
-
Patent No. :
201841006678
Filed :
13-02-2018
Published :
27-09-2019
Published
Greener synthesis of indolizine compounds
Sandeep C
Basavaraj Padmashali and Rashmi S. Kulkarni
-
Patent No. :
359559
Filed :
09-10-2015
Published :
17-03-2017
Granted
Scholarly Publications
1,2,3-Triazolyl-tetrahydropyrimidine Conjugates as Potential Sterol Carrier Protein-2 Inhibitors: Larvicidal Activity against the Malaria Vector <i>Anopheles arabiensis</i> and In Silico Molecular Docking Study
Open Access
Synthesis, crystal structure and Hirshfeld surface analysis of the hydrated form of N’, N-(1,4-phenylenebis(methanylylidene) di(iso-nicotinic hydrazide)
Anti-tubercular activity and molecular docking studies of indolizine derivatives targeting mycobacterial InhA enzyme
Open Access1-[4-bromo-2-(trifluoromethoxy)phenyl]-3-methyl-1H-1,2,4-triazole
Open AccessNucleophilic sulfur controlled efficient ketothioamide synthesis from tribromomethyl carbinols
Crystallography, molecular modeling, and cox-2 inhibition studies on indolizine derivatives
Open AccessSynthesis, crystal structure and Hirshfeld surface analysis of 2-(4-fluorophenyl)-2,3–dihydroquinazolin-4(1H)-one
Novel series of methyl 3-(Substituted benzoyl)-7-substituted-2-phenylindolizine-1-carboxylates as promising anti-inflammatory agents: Molecular modeling studies
Open Access
Showing 1 to 8 of 167 publications